Table 2. Pharmacological management of multi-drug resistant (MDR) tuberculosis (TB)
First-line oral drugsInjectable bactericidal drugs#Fluoroquinolones#Second-line bacteriostatic drugsOther drugs with unclear or unproven efficacy
RifampicinStreptomycinMoxifloxacinCycloserineClofazimine
IsoniazidAmikacinGatifloxacinp-aminosalicyclic acidClarithromycin
RifabutinKanamycinOfloxacinProthionamideAmoxicillin/clavulanate
EthanmbutolCapreomycinLevofloxacinEthionamideLinezolid
PyrizinamideTerizidoneImipenem/cilastatin
Thioacetazone
High-dose isoniazid
Order in which drugs are added to MDR-TB regimen →
  • #: all MDR-TB regimens should include one injectable and one fluoroquinolone where possible; : by definition, isolates classed as MDR will be resistant to these drugs.